BERARDINELLI, DILETTA
BERARDINELLI, DILETTA
Dipartimento Scienze Biomediche e Sanita' Pubblica
3-CMC, 4-CMC, and 4-BMC Human Metabolic Profiling: New Major Pathways to Document Consumption of Methcathinone Analogues?
2024-01-01 Berardinelli, Diletta; Taoussi, Omayema; Daziani, Gloria; Tavoletta, Francesco; Ricci, Giovanna; Tronconi, Livio P.; Adamowicz, Piotr; Busardo, Francesco Paolo; Carlier, Jeremy
3F-α-pyrrolydinovalerophenone (3F-α-PVP) in vitro human metabolism: Multiple in silico predictions to assist in LC-HRMS/MS analysis and targeted/untargeted data mining
2022-01-01 Carlier, J.; Berardinelli, D.; Montanari, E.; Sirignano, A.; Di Trana, A.; Busardo, F. P.
A new UHPLC-MS/MS method to assess cannabidiol and Δ9-tetrahydrocannabinol and respective metabolites in hair. Application to patients treated with medical cannabis|Sviluppo e validazione di un nuovo metodo in UHPLC-MS/MS per la determinazione di cannabidiolo e di tetraidrocannabinolo e relativi metaboliti in matrice pilifera. Applicazione su pazienti trattati con cannabis medica
2022-01-01 Faro, A. F. L.; Berardinelli, D.; Di Muzio, M. M.; Berretta, P.; Tini, A.
Comparison of authentic urine N-ethylpentedrone metabolites to predicted in silico and in vitro human hepatocyte metabolism
2025-01-01 Daziani, Gloria; Taoussi, Omayema; Berardinelli, Diletta; Bambagiotti, Giulia; Huestis, Marilyn A.; Busardo', Francesco P.; Carlier, Jeremy
Development of a novel enantioselective high-performance liquid chromatography–mass spectrometry method for the differentiation of dextro- and levo-methorphan and their O-demethylated metabolites in human blood and its application to post-mortem samples
2024-01-01 Jorbenadze, Saba; Khatiashvili, Tamar; Chelidze, Aluda; Lo Faro, Alfredo Fabrizio; Farkas, Tivadar; Tini, Anastasio; Sprega, Giorgia; Berardinelli, Diletta; Busardo, Francesco Paolo; Chankvetadze, Bezhan
Development of an enantioselective high-performance liquid chromatography-tandem mass spectrometry method for the quantitative determination of methorphan and its O-demethylated metabolite in human blood and its application to post-mortem samples
2023-01-01 Lo Faro, Alfredo Fabrizio; Berardinelli, Diletta; Sprega, Giorgia; Tini, Anastasio; Carlier, Jeremy; Farkas, Tivadar; Busardo', Francesco Paolo; Chankvetadze, Bezhan
Development of enantioselective high-performance liquid chromatography-tandem mass spectrometry method for quantitative determination of methylone and some of its metabolites in oral fluid
2023-01-01 Lo Faro, Alfredo Fabrizio; Sprega, Giorgia; Berardinelli, Diletta; Tini, Anastasio; Poyatos, Lourdes; Pichini, Simona; Farrè, Magì; Farkas, Tivadar; Busardo', Francesco Paolo; Giunashvili, Lasha; Chankvetadze, Bezhan
Development of enantioselective high-performance liquid chromatography-tandem mass spectrometry method for the quantitative determination of 3,4-methylenedioxy-methamphetamine (MDMA) and its phase-1 metabolites in human biological fluids
2024-01-01 Lo Faro, Alfredo Fabrizio; Sprega, Giorgia; Poyatos, Lourdes; Papaseit, Esther; Berretta, Paolo; Di Giorgi, Alessandro; Farre, Magì; Takaishvili, Nino; Farkas, Tivadar; Busardo, Francesco Paolo; Chankvetadze, Bezhan; Berardinelli, Diletta; Tini, Anastasio
Dipyanone, a new methadone-like synthetic opioid: In vitro and in vivo human metabolism and pharmacological profiling
2025-01-01 Berardinelli, Diletta; Kutzler, Johannes; Taoussi, Omayema; Zaami, Simona; Pichini, Simona; Basile, Giuseppe; Busardo', Francesco Paolo; Auwärter, Volker; Carlier, Jeremy
Exploring the Metabolism of Flubrotizolam, a Potent Thieno-Triazolo Diazepine, Using Human Hepatocytes and High-Resolution Mass Spectrometry
2024-01-01 Gameli, Prince Sellase; Kutzler, Johannes; Berardinelli, Diletta; Carlier, Jeremy; Auwärter, Volker; Busardò, Francesco Paolo
Human metabolism and basic pharmacokinetic evaluation of AP-238: A recently emerged acylpiperazine opioid
2023-01-01 Brunetti, Pietro; Berardinelli, Diletta; Giorgetti, Arianna; Schwelm, Hannes Max; Haschimi, Belal; Pelotti, Susi; Busardo', Francesco Paolo; Auwärter, Volker
Human metabolism and pharmacological profiling of protonitazepyne and metonitazepyne, two highly potent nitazenes: prediction of main metabolite activity based on µ-opioid receptor docking simulations
2025-01-01 Berardinelli, Diletta; Taoussi, Omayema; Ovat, Duygu Yeşim; Pichini, Simona; Pulver, Benedikt; Auwärter, Volker; Busardò, Francesco Paolo; Basile, Giuseppe; Laudadio, Emiliano; Carlier, Jeremy
Human metabolism of four synthetic benzimidazole opioids: isotonitazene, metonitazene, etodesnitazene, and metodesnitazene
2024-01-01 Taoussi, Omayema; Berardinelli, Diletta; Zaami, Simona; Tavoletta, Francesco; Basile, Giuseppe; Kronstrand, Robert; Auwärter, Volker; Busardò, Francesco P.; Carlier, Jeremy
In silico and in vitro human metabolism of IOX2, a performance-enhancing doping agent
2024-01-01 Taoussi, Omayema; Gameli, Prince Sellase; Berardinelli, Diletta; Busardò, Francesco Paolo; Tini, Anastasio; Carlier, Jeremy
In Vitro Metabolism of a Benzofuran-Substituted Nitazene: Ethyleneoxynitazene
2025-01-01 Taoussi, Omayema; Ovat, Duygu Yeşim; Tavoletta, Francesco; Tini, Anastasio; Bambagiotti, Giulia; Carlier, Jeremy; Auwärter, Volker; Busardo', Francesco Paolo; Berardinelli, Diletta
In vitro, in vivo metabolism and quantification of the novel synthetic opioid N-piperidinyl etonitazene (etonitazepipne)
2024-01-01 Berardinelli, Diletta; Taoussi, Omayema; Carlier, Jeremy; Tini, Anastasio; Zaami, Simona; Sundermann, Tom; Busardò, Francesco Paolo; Auwärter, Volker
In vivo and in vitro metabolism of the designer benzodiazepine, bretazenil: a comparison of pooled human hepatocytes and liver microsomes with postmortem urine and blood samples
2025-01-01 Gameli, Prince S.; Kutzler, Johannes; Huppertz, Laura M.; Berardinelli, Diletta; Tronconi, Livio; Basile, Giuseppe; Carlier, Jeremy; Busardo', Francesco P.; Auwärter, Volker
Liquid chromatography in forensic toxicology
2023-01-01 Berardinelli, Diletta; Tini, Anastasio; Montanari, Eva; Berretta, Paolo; Di Trana, Annagiulia
Metabolism and Pharmacological Characterization at μ-, κ-, and δ- Opioid Receptors Using a Novel Non-Radioactive Assay of Nitazenes and Methadone-like Synthetic Opioids
2025-03-31 Berardinelli, Diletta
Methylone and MDMA Pharmacokinetics Following Controlled Administration in Humans
2022-01-01 Poyatos, Lourdes; Lo Faro, Alfredo Fabrizio Francesco; Berardinelli, Diletta; Sprega, Giorgia; Malaca, Sara; Pichini, Simona; Huestis, Marilyn A.; Papaseit, Esther; Pérez-Mañá, Clara; Busardo', Francesco Paolo; Farré, Magí
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 3-CMC, 4-CMC, and 4-BMC Human Metabolic Profiling: New Major Pathways to Document Consumption of Methcathinone Analogues? | 1-gen-2024 | Berardinelli, Diletta; Taoussi, Omayema; Daziani, Gloria; Tavoletta, Francesco; Ricci, Giovanna; Tronconi, Livio P.; Adamowicz, Piotr; Busardo, Francesco Paolo; Carlier, Jeremy | |
| 3F-α-pyrrolydinovalerophenone (3F-α-PVP) in vitro human metabolism: Multiple in silico predictions to assist in LC-HRMS/MS analysis and targeted/untargeted data mining | 1-gen-2022 | Carlier, J.; Berardinelli, D.; Montanari, E.; Sirignano, A.; Di Trana, A.; Busardo, F. P. | |
| A new UHPLC-MS/MS method to assess cannabidiol and Δ9-tetrahydrocannabinol and respective metabolites in hair. Application to patients treated with medical cannabis|Sviluppo e validazione di un nuovo metodo in UHPLC-MS/MS per la determinazione di cannabidiolo e di tetraidrocannabinolo e relativi metaboliti in matrice pilifera. Applicazione su pazienti trattati con cannabis medica | 1-gen-2022 | Faro, A. F. L.; Berardinelli, D.; Di Muzio, M. M.; Berretta, P.; Tini, A. | |
| Comparison of authentic urine N-ethylpentedrone metabolites to predicted in silico and in vitro human hepatocyte metabolism | 1-gen-2025 | Daziani, Gloria; Taoussi, Omayema; Berardinelli, Diletta; Bambagiotti, Giulia; Huestis, Marilyn A.; Busardo', Francesco P.; Carlier, Jeremy | |
| Development of a novel enantioselective high-performance liquid chromatography–mass spectrometry method for the differentiation of dextro- and levo-methorphan and their O-demethylated metabolites in human blood and its application to post-mortem samples | 1-gen-2024 | Jorbenadze, Saba; Khatiashvili, Tamar; Chelidze, Aluda; Lo Faro, Alfredo Fabrizio; Farkas, Tivadar; Tini, Anastasio; Sprega, Giorgia; Berardinelli, Diletta; Busardo, Francesco Paolo; Chankvetadze, Bezhan | |
| Development of an enantioselective high-performance liquid chromatography-tandem mass spectrometry method for the quantitative determination of methorphan and its O-demethylated metabolite in human blood and its application to post-mortem samples | 1-gen-2023 | Lo Faro, Alfredo Fabrizio; Berardinelli, Diletta; Sprega, Giorgia; Tini, Anastasio; Carlier, Jeremy; Farkas, Tivadar; Busardo', Francesco Paolo; Chankvetadze, Bezhan | |
| Development of enantioselective high-performance liquid chromatography-tandem mass spectrometry method for quantitative determination of methylone and some of its metabolites in oral fluid | 1-gen-2023 | Lo Faro, Alfredo Fabrizio; Sprega, Giorgia; Berardinelli, Diletta; Tini, Anastasio; Poyatos, Lourdes; Pichini, Simona; Farrè, Magì; Farkas, Tivadar; Busardo', Francesco Paolo; Giunashvili, Lasha; Chankvetadze, Bezhan | |
| Development of enantioselective high-performance liquid chromatography-tandem mass spectrometry method for the quantitative determination of 3,4-methylenedioxy-methamphetamine (MDMA) and its phase-1 metabolites in human biological fluids | 1-gen-2024 | Lo Faro, Alfredo Fabrizio; Sprega, Giorgia; Poyatos, Lourdes; Papaseit, Esther; Berretta, Paolo; Di Giorgi, Alessandro; Farre, Magì; Takaishvili, Nino; Farkas, Tivadar; Busardo, Francesco Paolo; Chankvetadze, Bezhan; Berardinelli, Diletta; Tini, Anastasio | |
| Dipyanone, a new methadone-like synthetic opioid: In vitro and in vivo human metabolism and pharmacological profiling | 1-gen-2025 | Berardinelli, Diletta; Kutzler, Johannes; Taoussi, Omayema; Zaami, Simona; Pichini, Simona; Basile, Giuseppe; Busardo', Francesco Paolo; Auwärter, Volker; Carlier, Jeremy | |
| Exploring the Metabolism of Flubrotizolam, a Potent Thieno-Triazolo Diazepine, Using Human Hepatocytes and High-Resolution Mass Spectrometry | 1-gen-2024 | Gameli, Prince Sellase; Kutzler, Johannes; Berardinelli, Diletta; Carlier, Jeremy; Auwärter, Volker; Busardò, Francesco Paolo | |
| Human metabolism and basic pharmacokinetic evaluation of AP-238: A recently emerged acylpiperazine opioid | 1-gen-2023 | Brunetti, Pietro; Berardinelli, Diletta; Giorgetti, Arianna; Schwelm, Hannes Max; Haschimi, Belal; Pelotti, Susi; Busardo', Francesco Paolo; Auwärter, Volker | |
| Human metabolism and pharmacological profiling of protonitazepyne and metonitazepyne, two highly potent nitazenes: prediction of main metabolite activity based on µ-opioid receptor docking simulations | 1-gen-2025 | Berardinelli, Diletta; Taoussi, Omayema; Ovat, Duygu Yeşim; Pichini, Simona; Pulver, Benedikt; Auwärter, Volker; Busardò, Francesco Paolo; Basile, Giuseppe; Laudadio, Emiliano; Carlier, Jeremy | |
| Human metabolism of four synthetic benzimidazole opioids: isotonitazene, metonitazene, etodesnitazene, and metodesnitazene | 1-gen-2024 | Taoussi, Omayema; Berardinelli, Diletta; Zaami, Simona; Tavoletta, Francesco; Basile, Giuseppe; Kronstrand, Robert; Auwärter, Volker; Busardò, Francesco P.; Carlier, Jeremy | |
| In silico and in vitro human metabolism of IOX2, a performance-enhancing doping agent | 1-gen-2024 | Taoussi, Omayema; Gameli, Prince Sellase; Berardinelli, Diletta; Busardò, Francesco Paolo; Tini, Anastasio; Carlier, Jeremy | |
| In Vitro Metabolism of a Benzofuran-Substituted Nitazene: Ethyleneoxynitazene | 1-gen-2025 | Taoussi, Omayema; Ovat, Duygu Yeşim; Tavoletta, Francesco; Tini, Anastasio; Bambagiotti, Giulia; Carlier, Jeremy; Auwärter, Volker; Busardo', Francesco Paolo; Berardinelli, Diletta | |
| In vitro, in vivo metabolism and quantification of the novel synthetic opioid N-piperidinyl etonitazene (etonitazepipne) | 1-gen-2024 | Berardinelli, Diletta; Taoussi, Omayema; Carlier, Jeremy; Tini, Anastasio; Zaami, Simona; Sundermann, Tom; Busardò, Francesco Paolo; Auwärter, Volker | |
| In vivo and in vitro metabolism of the designer benzodiazepine, bretazenil: a comparison of pooled human hepatocytes and liver microsomes with postmortem urine and blood samples | 1-gen-2025 | Gameli, Prince S.; Kutzler, Johannes; Huppertz, Laura M.; Berardinelli, Diletta; Tronconi, Livio; Basile, Giuseppe; Carlier, Jeremy; Busardo', Francesco P.; Auwärter, Volker | |
| Liquid chromatography in forensic toxicology | 1-gen-2023 | Berardinelli, Diletta; Tini, Anastasio; Montanari, Eva; Berretta, Paolo; Di Trana, Annagiulia | |
| Metabolism and Pharmacological Characterization at μ-, κ-, and δ- Opioid Receptors Using a Novel Non-Radioactive Assay of Nitazenes and Methadone-like Synthetic Opioids | 31-mar-2025 | Berardinelli, Diletta | |
| Methylone and MDMA Pharmacokinetics Following Controlled Administration in Humans | 1-gen-2022 | Poyatos, Lourdes; Lo Faro, Alfredo Fabrizio Francesco; Berardinelli, Diletta; Sprega, Giorgia; Malaca, Sara; Pichini, Simona; Huestis, Marilyn A.; Papaseit, Esther; Pérez-Mañá, Clara; Busardo', Francesco Paolo; Farré, Magí |