Sfoglia per Autore
Synthesis of Enantiomerically Pure 3-Amino-2-methylenealkanoates (Aza-Morita–Baylis–Hillman Adducts) Mediated by Cinchona Alkaloids
2011-01-01 Martelli, G.; Orena, Mario; Rinaldi, Samuele
A Bifunctional β-Isocupreidine Derivative as Catalyst for the EnantioselectiveMorita–Baylis–Hillman Reaction and a Mechanistic Rationale forEnantioselectivity
2012-01-01 Martelli, Gianluca; Orena, Mario; Rinaldi, Samuele
Ammonolysis of morpholine-2,5-diones: participation of the primary amide group. Part 2
2012-01-01 Arcelli, A.; Bongini, A.; Porzi, G.; Rinaldi, Samuele
beta-Peptoids: synthesis of a novel dimer having a fully extendedconformation
2012-01-01 Martelli, Gianluca; Monsignori, Antonella; Orena, Mario; Rinaldi, Samuele; Castellucci, N.; Tomasini, C. .
Stereoselective alkylation of chiral pyrrolidin-2-ones leading to novel conformationally restricted analogues of 3-methylaspartic acid: a computational investigation
2012-01-01 Galeazzi, Roberta; Martelli, G.; Orena, Mario; Rinaldi, Samuele
Analogues of nucleosides: synthesis of chiral pyrrolidin-2-ones or pyrrolidines-bearing nucleobases
2014-01-01 Martelli, Gianluca; Monsignori, Antonella; Orena, Mario; Rinaldi, Samuele
Recent Advances in Chemistry of γ-Lactams: Part I. Synthesis Starting from Acyclic or Cyclic Precursors
2014-01-01 Martelli, Gianluca; Orena, Mario; Rinaldi, Samuele
Recent Advances in Chemistry of γ-Lactams: Part II. Functionalization by C-C or C-Heteroatom Bond Formation
2014-01-01 Martelli, Gianluca; Monsignori, Antonella; Orena, Mario; Rinaldi, Samuele
Synthesis of a cyclic isostere of α-methyl homoserine by a stereoselective acylation–alkylation sequence of a chiral γ-lactam
2014-01-01 Civitavecchia, Annafelicia; Martelli, Gianluca; Orena, Mario; Rinaldi, Samuele
Novel nucleoside analogs tethered on (3R,4R)-4-(hydroxymethyl)pyrrolidin-3-ol
2015-01-01 Amici, Adolfo; Martelli, Gianluca; Orena, Mario; Rinaldi, Samuele
Highly stable atropisomers by electrophilic amination of a chiral γ-lactam within the synthesis of an elusive conformationally restricted analogue of α-methylhomoserine
2016-01-01 Amabili, Paolo; Amici, Adolfo; Civitavecchia, Annafelicia; Maggiore, Beatrice; Orena, Mario; Rinaldi, Samuele; Tolomelli, Alessandra
Synthesis of Enantiopure Isosteres of Amino Acids Containing a Quaternary Stereocenter: Experimental and Computational Evaluation of a Novel Class of Atropisomers
2018-01-01 Amabili, Paolo; Amici, Adolfo; Campisi, Giovanni; Guerra, Giulia; Monari, Magda; Orena, Mario; Piccinelli, Fabio; Rinaldi, Samuele; Tolomelli, Alessandra
Imidazolidinone-Tethered α-Hydrazidopeptides – Synthesis and Conformational Investigation
2018-01-01 Amabili, Paolo; Calvaresi, Matteo; Martelli, Gianluca; Orena, Mario; Rinaldi, Samuele; Sgolastra, Federica
Synthesis, structural insights and activity of different classes of biomolecules
2020-01-01 Giorgini, E.; Biavasco, F.; Galeazzi, R.; Gioacchini, G.; Giovanetti, E.; Mobbili, G.; Orena, M.; Ortore, M. G.; Rinaldi, S.; Scire, A. A.; Spinozzi, F.; Tanfani, F.; Vignaroli, C.; Mariani, P.
Simple amphiphilic α-hydrazido acids: Rational design, synthesis, and in vitro bioactivity profile of a novel class of potential antimicrobial compounds
2020-01-01 Amabili, P.; Biavasco, F.; Brenciani, A.; Citterio, B.; Corbisiero, D.; Ferrazzano, L.; Fioriti, S.; Guerra, G.; Orena, M.; Rinaldi, S.
The diverse world of foldamers: Endless possibilities of self-assembly
2020-01-01 Rinaldi, S.
Identification of a novel nitroflavone-based scaffold for designing mutant-selective EGFR tyrosine kinase inhibitors targeting T790M and C797S resistance in advanced NSCLC
2022-01-01 Minnelli, Cristina; Laudadio, Emiliano; Sorci, Leonardo; Sabbatini, Giulia; Galeazzi, Roberta; Amici, Adolfo; Semrau, Marta S.; Storici, Paola; Rinaldi, Samuele; Stipa, Pierluigi; Marcaccio, Massimo; Mobbili, Giovanna
Asymmetric Construction of γ-lactams Displaying All-carbon, Aza-, Thia- and Oxa-quaternary Chiral Centers
2023-01-01 Orena, Mario; Rinaldi, Samuele
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